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BPS Bioscience Inc.
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當(dāng)前位置:BPS Bioscience Inc.>>Inhibitors / Activators>> 27023SP600125

SP600125

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產(chǎn)品型號(hào)27023

品       牌BPS Bioscience

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更新時(shí)間:2023-12-19 22:39:17瀏覽次數(shù):108次

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●Purchase●DescriptionNovel,potentandselectiveJNK-1,-2,and-3inhibitor(Ki=0
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Description

Novel, potent and selective JNK-1,-2, and -3 inhibitor (Ki = 0.19 µM). SP600125 is an ATP-competitive reversible inhibitor with >20-fold selectivity vs. a range of kinases and enzymes tested. In cells, SP600125 caused a dose-dependent inhibition of the phosphorylation of c-Jun, the expression of inflammatory genes IL-2, COX-2, TNF-α, IFN-γ, and blocked the activation and differentiation of primary human CD4 cell cultures.

Synonyms
Anthra(1,9-cd)pyrazol-6(2H)-one, 1,9-Pyrazoloanthrone, Anthrapyrazolone, JNK Inhibitor II

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